PF-00562271抑制劑PF-562271 (besylate) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM, ~10-fold less potent for Pyk2 than FAK and >100-fold selectivity against other protein kinases, except for some CDKs.
產品名稱: | PF-00562271 | ||
英文名: | PF-562271 besylate | ||
CAS NO.: | 939791-38-5 | ||
分子式: | C27H26F3N7O6S2 | ||
分子量: | 665.663853168488 | ||
產品品牌: | targetmol | ||
產品規格: | 1mg |