沙普替尼抑制劑AZD8931, a reversible, ATP competitive inhibitor of EGFR(IC50=4 nM), ErbB2(IC50=3 nM) and ErbB3(IC50=4 nM), is more effective over Gefitinib or Lapatinib against NSCLC cell, 100-fold more specific for the ErbB family over MNK1 and Flt.
產品名稱: | 沙普替尼 | ||
英文名: | Sapitinib | ||
CAS NO.: | 848942-61-0 | ||
分子式: | C23H25ClFN5O3 | ||
分子量: | 473.927707433701 | ||
產品品牌: | targetmol | ||
產品規格: | 1mg |